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Readily Available Chiral Benzimidazoles-Derived Guanidines as Organocatalysts in the Asymmetric α-Amination of 1,3-Dicarbonyl Compounds

The synthesis and the evaluation as organocatalysts of new chiral guanidines derived from benzimidazoles in the enantioselective α-amination of 1,3-dicarbonyl compounds using di-t-butylazodicarboxylate as aminating agent is herein disclosed. The catalysts are readily synthesized through the reaction...

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Detalles Bibliográficos
Autores principales:	Benavent, Llorenç, Puccetti, Francesco, Baeza, Alejandro, Gómez-Martínez, Melania
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2017
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6152235/ https://www.ncbi.nlm.nih.gov/pubmed/28800100 http://dx.doi.org/10.3390/molecules22081333

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