Suzuki-Type Cross-Coupling Reaction of Unprotected 3-Iodoindazoles with Pinacol Vinyl Boronate: An Expeditive C-3 Vinylation of Indazoles under Microwave Irradiation

Herein we report an expeditive C-3 vinylation of unprotected 3-iodoindazoles under microwave irradiation. Ten C-5 substituted 3-vinylindazole derivatives, nine of them novel, were synthesized through this method, which proceeds in moderate to excellent yields starting from C-5 substituted 3-iodoinda...

Descripción completa

Detalles Bibliográficos
Autores principales: Vera, Gonzalo, Diethelm, Benjamín, Terraza, Claudio A., Recabarren-Gajardo, Gonzalo
Formato: Online Artículo Texto
Lenguaje:English
Publicado: MDPI 2018
Materias:
Communication
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6222620/
https://www.ncbi.nlm.nih.gov/pubmed/30115838
http://dx.doi.org/10.3390/molecules23082051

Internet

https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6222620/
https://www.ncbi.nlm.nih.gov/pubmed/30115838
http://dx.doi.org/10.3390/molecules23082051

Ejemplares similares