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Preparation and Properties of New Co-Crystals of Ibandronate with Gluco- or Galactopyranoside Derivatives †

Mixtures of ibandronate monosodium salt with eleven gluco- and/or galacto-pyranoside derivatives as counterions were designed to prepare co-crystals with improved intestinal absorption. In general, gastrointestinal absorption of bisphosphonates after oral administration is approximately 1%. Co-cryst...

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Detalles Bibliográficos
Autores principales: Oktabec, Zbynek, Kos, Jiri, Mandelova, Zuzana, Havelkova, Lenka, Pekarek, Tomas, Rezacova, Anna, Placek, Lukas, Tkadlecova, Marcela, Havlicek, Jaroslav, Dohnal, Jiri, Jampílek, Josef
Formato: Online Artículo Texto
Lenguaje:English
Publicado: MDPI 2010
Materias:
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6259308/
https://www.ncbi.nlm.nih.gov/pubmed/21150819
http://dx.doi.org/10.3390/molecules15128973