Cargando…

Design, Synthesis and the Biological Evaluation of New 1,3-Thiazolidine-4-ones Based on the 4-Amino-2,3-dimethyl-1-phenyl-3-pyrazolin-5-one Scaffold

New thiazolidine-4-one derivatives based on the 4-aminophenazone (4-amino-2,3-dimethyl-1-phenyl-3-pyrazolin-5-one) scaffold have been synthesized as potential anti-inflammatory drugs. The pyrazoline derivatives are known especially for their antipyretic, analgesic and anti-inflammatory effects, but...

Descripción completa

Detalles Bibliográficos
Autores principales:	Apotrosoaei, Maria, Vasincu, Ioana Mirela, Dragan, Maria, Buron, Frédéric, Routier, Sylvain, Profire, Lenuta
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2014
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6270961/ https://www.ncbi.nlm.nih.gov/pubmed/25255761 http://dx.doi.org/10.3390/molecules190913824

Ejemplares similares

Synthesis and Biological Evaluation of New 1,3-Thiazolidine-4-one Derivatives of 2-(4-Isobutylphenyl)propionic Acid
por: Vasincu, Ioana Mirela, et al.
Publicado: (2014)

Synthesis and biological evaluation of the new 1,3-dimethylxanthine derivatives with thiazolidine-4-one scaffold
por: Constantin, Sandra, et al.
Publicado: (2017)

Synthesis and biological evaluation of new 1,3-thiazolidine-4-one derivatives of nitro-l-arginine methyl ester
por: Pânzariu, Andreea-Teodora, et al.
Publicado: (2016)

New ibuprofen derivatives with thiazolidine-4-one scaffold with improved pharmaco-toxicological profile
por: Vasincu, Ioana-Mirela, et al.
Publicado: (2021)

Formulation and Characterization of New Polymeric Systems Based on Chitosan and Xanthine Derivatives with Thiazolidin-4-One Scaffold
por: Constantin, Sandra Madalina, et al.
Publicado: (2019)

Complexes of Ibuprofen Thiazolidin-4-One Derivatives with β-Cyclodextrin: Characterization and In Vivo Release Profile and Biological Evaluation
por: Vasincu, Ioana Mirela, et al.
Publicado: (2023)

The Synthesis and the Biological Evaluation of New Thiazolidin-4-one Derivatives Containing a Xanthine Moiety
por: Lupascu, Florentina Geanina, et al.
Publicado: (2013)

3-Phenyl-2-thioxo-1,3-thiazolidin-4-one
por: Zhu, Feng-Xia, et al.
Publicado: (2008)

3-Benzyl-2-phenyl-1,3-thiazolidin-4-one
por: Fun, Hoong-Kun, et al.
Publicado: (2011)

5-Benzylidene-3-phenyl-2-phenylimino-1,3-thiazolidin-4-one
por: Zeller, Matthias, et al.
Publicado: (2011)

Synthesis of novel series of 3,5-disubstituted imidazo[1,2-d] [1,2,4]thiadiazoles involving S(N)Ar and Suzuki–Miyaura cross-coupling reactions
por: Pescheteau, Clémentine, et al.
Publicado: (2022)

(5S)-5-Methyl-3-phenyl-2-sulfanylidene-1,3-thiazolidin-4-one
por: Jiang, Jun-Rong, et al.
Publicado: (2011)

2,3-Diphenyl-1,3-thiazolidin-4-one
por: Yennawar, Hemant P., et al.
Publicado: (2014)

4-(4-Bromophenylhydrazono)-1-(5-bromopyrimidin-2-yl)-3-methyl-2-pyrazolin-5-one
por: Subramanyam, M., et al.
Publicado: (2008)

(Z)-3-(2-Hydroxyethyl)-2-(phenylimino)-1,3-thiazolidin-4-one
por: Mohamed, Shaaban K., et al.
Publicado: (2012)

Design, Synthesis, In Silico and In Vitro Studies for New Nitric Oxide-Releasing Indomethacin Derivatives with 1,3,4-Oxadiazole-2-thiol Scaffold
por: Sava, Alexandru, et al.
Publicado: (2021)

Recent Biomedical Approaches for Chitosan Based Materials as Drug Delivery Nanocarriers
por: Iacob, Andreea Teodora, et al.
Publicado: (2021)

3-Cyclohexyl-2-thioxo-1,3-thiazolidin-4-one
por: Shahwar, Durre, et al.
Publicado: (2009)

3-Benzyl-2-sulfanylidene-1,3-thiazolidin-4-one
por: Shahwar, Durre, et al.
Publicado: (2010)

Facile synthesis, antimicrobial and antiviral evaluation of novel substituted phenyl 1,3-thiazolidin-4-one sulfonyl derivatives
por: Mandal, Milan Kumar, et al.
Publicado: (2021)

3-(4-Methylphenyl)-2-thioxo-1,3-thiazolidin-4-one
por: Shahwar, Durre, et al.
Publicado: (2010)

(5Z)-5-(2-Methylbenzylidene)-3-phenyl-2-thioxo-1,3-thiazolidin-4-one
por: Shahwar, Durre, et al.
Publicado: (2009)

(5Z)-5-(2-Hydroxybenzylidene)-3-phenyl-2-thioxo-1,3-thiazolidin-4-one
por: Shahwar, Durre, et al.
Publicado: (2009)

3,3-Dimethyl-9-phenyl-3,4-dihydroacridin-1(2H)-one
por: Ghorbani, Hosein, et al.
Publicado: (2008)

Crystal structure of a 1:1 adduct of triphenyltin chloride with 3-cyclohexhyl-2-phenyl-1,3-thiazolidin-4-one
por: Yennawar, Hemant P., et al.
Publicado: (2019)

1,4-Dimethyl-3-phenyl-3H-pyrazolo[3,4-c]isoquinolin-5(4H)-one
por: Meneghetti, Fiorella, et al.
Publicado: (2008)

Crystal structures of 2,3-bis(4-chlorophenyl)-1,3-thiazolidin-4-one and trans-2,3-bis(4-chlorophenyl)-1,3-thiazolidin-4-one 1-oxide
por: Yennawar, Hemant P., et al.
Publicado: (2015)

3-Butyl-2-phenyl-1,3-thiazolidine-1,4-dione
por: Wang, Qiang, et al.
Publicado: (2010)

3-[4-(Dimethylamino)phenyl]-1-(3-pyridyl)prop-2-en-1-one
por: Jayarama, A., et al.
Publicado: (2009)

3-(3-Methylphenyl)-2-thioxo-1,3-thiazolidin-4-one
por: Shahwar, Durre, et al.
Publicado: (2009)

3-Benzyl-2-(furan-2-yl)-1,3-thiazolidin-4-one
por: Fun, Hoong-Kun, et al.
Publicado: (2011)

(Z)-3-Benzyl-2-[(2-phenylcyclohex-2-enyl)imino]-1,3-thiazolidin-4-one
por: Ooi, Chin Wei, et al.
Publicado: (2012)

2-(4-Chlorophenyl)-3-p-tolyl-1,3-thiazolidin-4-one
por: Sun, Xiao-Jun, et al.
Publicado: (2009)

1-Chloroacetyl-3,3-dimethyl-2,6-diphenylpiperidin-4-one
por: Kavitha, T., et al.
Publicado: (2008)

2-(2,4-Dichlorophenyl)-3-[5-(3,5-dimethylphenyl)-1,3,4-thiadiazol-2-yl]thiazolidin-4-one
por: Wan, Rong, et al.
Publicado: (2007)

Synthesis and Antioxidant Activity of Some New Coumarinyl-1,3-Thiazolidine-4-ones
por: Čačić, Milan, et al.
Publicado: (2010)

3,4-Dimethyl-1-phenylpyrano[2,3-c]pyrazol-6(1H)-one
por: Ahmad, Neman, et al.
Publicado: (2011)

3-Benzyl-5-benzylidene-2-sulfanylidene-1,3-thiazolidin-4-one
por: Shahwar, Durre, et al.
Publicado: (2011)

2-Imino-3-(2-nitrophenyl)-1,3-thiazolidin-4-one
por: Zia-ur-Rehman, Muhammad, et al.
Publicado: (2011)

3-(2-Methylphenyl)-2-thioxo-1,3-thiazolidin-4-one
por: Shahwar, Durre, et al.
Publicado: (2009)

Cannot write session to /tmp/vufind_sessions/sess_3bdumsm6gj8mv24irrav70nucf