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Synthesis, Antiphospholipase A(2), Antiprotease, Antibacterial Evaluation and Molecular Docking Analysis of Certain Novel Hydrazones
Some novel hydrazone derivatives 6a–o were synthesized from the key intermediate 4-Chloro-N-(2-hydrazinocarbonyl-phenyl)-benzamide 5 and characterized using IR, (1)H-NMR, (13)C-NMR, mass spectroscopy and elemental analysis. The inhibitory potential against two secretory phospholipase A(2) (sPLA(2)),...
Autores principales: | El-Sayed, Nahed N. E., Alafeefy, Ahmed M., Bakht, Mohammed A., Masand, Vijay H., Aldalbahi, Ali, Chen, Nan, Fan, Chunhai, Ben Bacha, Abir |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
MDPI
2016
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6272960/ https://www.ncbi.nlm.nih.gov/pubmed/27918459 http://dx.doi.org/10.3390/molecules21121664 |
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