Exploring 6-Azaindole and 7-Azaindole Rings for Developing Cannabinoid Receptor 1 Allosteric Modulators

Introduction and Objective: Org27569 is a prototypical allosteric modulator of the cannabinoid receptor 1 (CB(1)). It belongs to the indole-2-carboxamide scaffold and has been intensively investigated in pharmacology and in structure–activity relationship (SAR) studies. Although azaindoles are rare...

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Detalles Bibliográficos
Autores principales: Immadi, Sri Sujana, Dopart, Rachel, Wu, Zhixing, Fu, Boqiao, Kendall, Debra A., Lu, Dai
Formato: Online Artículo Texto
Lenguaje:English
Publicado: Mary Ann Liebert, Inc., publishers 2018
Materias:
Original Research
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6290480/
https://www.ncbi.nlm.nih.gov/pubmed/30547095
http://dx.doi.org/10.1089/can.2018.0046

Internet

https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6290480/
https://www.ncbi.nlm.nih.gov/pubmed/30547095
http://dx.doi.org/10.1089/can.2018.0046

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