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Exploring 6-Azaindole and 7-Azaindole Rings for Developing Cannabinoid Receptor 1 Allosteric Modulators

Introduction and Objective: Org27569 is a prototypical allosteric modulator of the cannabinoid receptor 1 (CB(1)). It belongs to the indole-2-carboxamide scaffold and has been intensively investigated in pharmacology and in structure–activity relationship (SAR) studies. Although azaindoles are rare...

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Detalles Bibliográficos
Autores principales:	Immadi, Sri Sujana, Dopart, Rachel, Wu, Zhixing, Fu, Boqiao, Kendall, Debra A., Lu, Dai
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Mary Ann Liebert, Inc., publishers 2018
Materias:	Original Research
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6290480/ https://www.ncbi.nlm.nih.gov/pubmed/30547095 http://dx.doi.org/10.1089/can.2018.0046

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