Cargando…
Microwave-Assisted Stereoselective Heterocyclization to Novel Ring d-fused Arylpyrazolines in the Estrone Series
Microwave-assisted syntheses of novel ring d-condensed 2-pyrazolines in the estrone series were efficiently carried out from steroidal α,β-enones and hydrazine derivatives. The ring-closure reaction of 16-benzylidene estrone 3-methyl ether with hydrazine in acetic acid resulted in a 2:1 diastereomer...
Autores principales: | Mótyán, Gergő, Molnár, Barnabás, Wölfling, János, Frank, Éva |
---|---|
Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
MDPI
2019
|
Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6384934/ https://www.ncbi.nlm.nih.gov/pubmed/30720767 http://dx.doi.org/10.3390/molecules24030569 |
Ejemplares similares
-
The first Pd-catalyzed Buchwald–Hartwig aminations at C-2 or C-4 in the estrone series
por: Bacsa, Ildikó, et al.
Publicado: (2018) -
Microwave-Assisted Synthesis of Bioactive Six-Membered Heterocycles and Their Fused Analogues
por: Driowya, Mohsine, et al.
Publicado: (2016) -
Microwave-assisted synthesis of biologically relevant steroidal 17-exo-pyrazol-5'-ones from a norpregnene precursor by a side-chain elongation/heterocyclization sequence
por: Mótyán, Gergő, et al.
Publicado: (2018) -
Microwave-Assisted Syntheses of Bioactive Seven-Membered, Macro-Sized Heterocycles and Their Fused Derivatives
por: Driowya, Mohsine, et al.
Publicado: (2016) -
Synthesis and Biological Evaluation of Triazolyl 13α-Estrone–Nucleoside Bioconjugates
por: Bodnár, Brigitta, et al.
Publicado: (2016)