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Novel alanine serine cysteine transporter 2 (ASCT2) inhibitors based on sulfonamide and sulfonic acid ester scaffolds
The neutral amino acid transporter alanine serine cysteine transporter 2 (ASCT2) belongs to the solute carrier 1 (SLC1) family of transport proteins and transports neutral amino acids, such as alanine and glutamine, into the cell in exchange with intracellular amino acids. This amino acid transport...
Autores principales: | Ndaru, Elias, Garibsingh, Rachel-Ann A., Shi, YueYue, Wallace, Evan, Zakrepine, Paul, Wang, Jiali, Schlessinger, Avner, Grewer, Christof |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Rockefeller University Press
2019
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6400523/ https://www.ncbi.nlm.nih.gov/pubmed/30718375 http://dx.doi.org/10.1085/jgp.201812276 |
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