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Practical, metal-free remote heteroarylation of amides via unactivated C(sp(3))–H bond functionalization

Development of practical methods for the production of multi-functionalized amides is one of the most important topics in both synthetic chemistry and drug discovery. Disclosed herein is a new, efficient, site-selective heteroarylation of amides via C(sp(3))–H bond functionalization. Amidyl radicals...

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Detalles Bibliográficos
Autores principales:	Tang, Nana, Wu, Xinxin, Zhu, Chen
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Royal Society of Chemistry 2019
Materias:	Chemistry
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6640195/ https://www.ncbi.nlm.nih.gov/pubmed/31391914 http://dx.doi.org/10.1039/c9sc02564b

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