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Molecular docking, synthesis, kinetics study, structure–activity relationship and ADMET analysis of morin analogous as Helicobacter pylori urease inhibitors

BACKGROUND: Urease are responsible for several pathogenic states in human as well as in animals and its inhibition is utmost urgent. Clinically used drugs are associated with many side effects; recently several researches have shown that flavonoids have good urease inhibition properties. Morin, a na...

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Detalles Bibliográficos
Autores principales: Kataria, Ritu, Khatkar, Anurag
Formato: Online Artículo Texto
Lenguaje:English
Publicado: Springer International Publishing 2019
Materias:
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6661831/
https://www.ncbi.nlm.nih.gov/pubmed/31384793
http://dx.doi.org/10.1186/s13065-019-0562-2