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Acyl‐Directed ortho‐Borylation of Anilines and C7 Borylation of Indoles using just BBr(3)

Indoles are privileged heterocycles found in many biologically active pharmaceuticals and natural products. However, the selective functionalization of the benzenoid moiety in indoles in preference to the more reactive pyrrolic unit is a significant challenge. Herein we report that N‐acyl directing...

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Detalles Bibliográficos
Autores principales: Iqbal, Saqib A., Cid, Jessica, Procter, Richard J., Uzelac, Marina, Yuan, Kang, Ingleson, Michael J.
Formato: Online Artículo Texto
Lenguaje:English
Publicado: John Wiley and Sons Inc. 2019
Materias:
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6856876/
https://www.ncbi.nlm.nih.gov/pubmed/31461213
http://dx.doi.org/10.1002/anie.201909786