TMSBr-Promoted Cascade Cyclization of ortho-Propynol Phenyl Azides for the Synthesis of 4-Bromo Quinolines and Its Applications

Difficult-to-access 4-bromo quinolines are constructed directly from easily prepared ortho-propynol phenyl azides using TMSBr as acid-promoter. The cascade transformation performs smoothly to generate desired products in moderate to excellent yields with good functional groups compatibility. Notably...

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Detalles Bibliográficos
Autores principales: Jin, Fengyan, Yang, Tao, Song, Xian-Rong, Bai, Jiang, Yang, Ruchun, Ding, Haixin, Xiao, Qiang
Formato: Online Artículo Texto
Lenguaje:English
Publicado: MDPI 2019
Materias:
Article
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6864654/
https://www.ncbi.nlm.nih.gov/pubmed/31694215
http://dx.doi.org/10.3390/molecules24213999

Internet

https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6864654/
https://www.ncbi.nlm.nih.gov/pubmed/31694215
http://dx.doi.org/10.3390/molecules24213999

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