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Mild and Practical Indole C2 Allylation by Allylboration of in situ Generated 3‐Chloroindolenines

C2 allylation of indole derivatives is a challenging but important transformation given the biological relevance of the products. Herein we report a selective C2 allylation strategy that proceeds via allylboration of in situ‐generated 3‐chloroindolenines. The reaction is mild, practical, and compati...

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Detalles Bibliográficos
Autores principales: Saya, Jordy M., van Wordragen, Ellen D. H., Orru, Romano V. A., Ruijter, Eelco
Formato: Online Artículo Texto
Lenguaje:English
Publicado: John Wiley and Sons Inc. 2019
Materias:
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6919337/
https://www.ncbi.nlm.nih.gov/pubmed/31894179
http://dx.doi.org/10.1002/ejoc.201801745