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Inhibition survey with phenolic compounds against the δ- and η-class carbonic anhydrases from the marine diatom thalassiosira weissflogii and protozoan Plasmodium falciparum

The inhibition of δ- and η-class carbonic anhydrases (CAs; EC 4.2.1.1) was poorly investigated so far. Only one δ-CA, TweCA from the diatom Thalassiosira weissflogii, and one η-CA, PfCA, from Plasmodium falciparum, have been cloned and characterised to date. To enrich δ- and η-CAs inhibition profile...

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Detalles Bibliográficos
Autores principales: Alissa, Siham A., Alghulikah, Hanan A., ALOthman, Zeid A., Osman, Sameh M., Del Prete, Sonia, Capasso, Clemente, Nocentini, Alessio, Supuran, Claudiu T.
Formato: Online Artículo Texto
Lenguaje:English
Publicado: Taylor & Francis 2019
Materias:
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6968676/
https://www.ncbi.nlm.nih.gov/pubmed/31856608
http://dx.doi.org/10.1080/14756366.2019.1706089