Diverse N-Substituted Azole-Containing Amino Acids as Building Blocks for Cyclopeptides

[Image: see text] The preparation of 16 oxazole- or thiazole-containing amino esters bearing a wide array of N-substitution is reported. These were accessed in 40–92% yield via an AgClO(4)-promoted substitution reaction between a primary amine and a chloromethyl-functionalized thiazole or oxazole. T...

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Detalles Bibliográficos
Autores principales: Motevalli, Somayeh, Nguyen, Michelle T., Tan, Jiacheng, Fuller, Amelia A.
Formato: Online Artículo Texto
Lenguaje:English
Publicado: American Chemical Society 2020
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6977196/
https://www.ncbi.nlm.nih.gov/pubmed/31984279
http://dx.doi.org/10.1021/acsomega.9b03682

Internet

https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6977196/
https://www.ncbi.nlm.nih.gov/pubmed/31984279
http://dx.doi.org/10.1021/acsomega.9b03682

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