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Diverse N-Substituted Azole-Containing Amino Acids as Building Blocks for Cyclopeptides
[Image: see text] The preparation of 16 oxazole- or thiazole-containing amino esters bearing a wide array of N-substitution is reported. These were accessed in 40–92% yield via an AgClO(4)-promoted substitution reaction between a primary amine and a chloromethyl-functionalized thiazole or oxazole. T...
| Autores principales: | , , , |
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| Formato: | Online Artículo Texto |
| Lenguaje: | English |
| Publicado: |
American Chemical Society
2020
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| Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6977196/ https://www.ncbi.nlm.nih.gov/pubmed/31984279 http://dx.doi.org/10.1021/acsomega.9b03682 |