Interaction of the Anti-Proliferative GPER Inverse Agonist ERα17p with the Breast Cancer Cell Plasma Membrane: From Biophysics to Biology

The peptide ERα17p, which corresponds to the 295-311 fragment of the hinge/AF2 domains of the human estrogen receptor α (ERα), exerts apoptosis in breast cancer cells through a mechanism involving the G protein-coupled estrogen-dependent receptor GPER. Besides this receptor-mediated mechanism, we ha...

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Detalles Bibliográficos
Autores principales: Trichet, Michaël, Lappano, Rosamaria, Belnou, Mathilde, Salazar Vazquez, Lilian Shadai, Alves, Isabel, Ravault, Delphine, Sagan, Sandrine, Khemtemourian, Lucie, Maggiolini, Marcello, Jacquot, Yves
Formato: Online Artículo Texto
Lenguaje:English
Publicado: MDPI 2020
Materias:
Article
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7072814/
https://www.ncbi.nlm.nih.gov/pubmed/32075246
http://dx.doi.org/10.3390/cells9020447

Internet

https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7072814/
https://www.ncbi.nlm.nih.gov/pubmed/32075246
http://dx.doi.org/10.3390/cells9020447

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