Cargando…

Structure-activity relationship studies of lipophilic teicoplanin pseudoaglycon derivatives as new anti-influenza virus agents

Six series of semisynthetic lipophilic glycopeptide antibiotic derivatives were evaluated for in vitro activity against influenza A and B viruses. The new teicoplanin pseudoaglycon-derived lipoglycopeptides were prepared by coupling one or two side chains to the N-terminus of the glycopeptide core,...

Descripción completa

Detalles Bibliográficos
Autores principales:	Szűcs, Zsolt, Kelemen, Viktor, Le Thai, Son, Csávás, Magdolna, Rőth, Erzsébet, Batta, Gyula, Stevaert, Annelies, Vanderlinden, Evelien, Naesens, Lieve, Herczegh, Pál, Borbás, Anikó
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Elsevier Masson SAS. 2018
Materias:	Research Paper
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7115582/ https://www.ncbi.nlm.nih.gov/pubmed/30170320 http://dx.doi.org/10.1016/j.ejmech.2018.08.058

Ejemplares similares

Synthesis of Antiviral Perfluoroalkyl Derivatives of Teicoplanin and Vancomycin
por: Bereczki, Ilona, et al.
Publicado: (2020)

Reprogramming of the Antibacterial Drug Vancomycin Results in Potent Antiviral Agents Devoid of Antibacterial Activity
por: Szűcs, Zsolt, et al.
Publicado: (2020)

The First Dimeric Derivatives of the Glycopeptide Antibiotic Teicoplanin
por: Bereczki, Ilona, et al.
Publicado: (2022)

Synthesis of an amphiphilic vancomycin aglycone derivative inspired by polymyxins: overcoming glycopeptide resistance in Gram-positive and Gram-negative bacteria in synergy with teicoplanin in vitro
por: Szűcs, Zsolt, et al.
Publicado: (2022)

Anti-influenza virus activity and structure–activity relationship of aglycoristocetin derivatives with cyclobutenedione carrying hydrophobic chains
por: Naesens, Lieve, et al.
Publicado: (2009)

Semisynthetic teicoplanin derivatives with dual antimicrobial activity against SARS-CoV-2 and multiresistant bacteria
por: Bereczki, Ilona, et al.
Publicado: (2022)

Photoinitiated Thiol−Ene Reactions of Various 2,3‐Unsaturated O‐, C‐ S‐ and N‐Glycosides – Scope and Limitations Study
por: Kelemen, Viktor, et al.
Publicado: (2020)

The Very First Modification of Pleuromutilin and Lefamulin by Photoinitiated Radical Addition Reactions—Synthesis and Antibacterial Studies
por: Thai Le, Son, et al.
Publicado: (2021)

Pseudoaglycone of Spinosyn A
por: Chai, Hongxin, et al.
Publicado: (2012)

The Influenza Virus Polymerase Complex: An Update on Its Structure, Functions, and Significance for Antiviral Drug Design
por: Stevaert, Annelies, et al.
Publicado: (2016)

Investigation of the Binding Affinity of a Broad Array of l-Fucosides with Six Fucose-Specific Lectins of Bacterial and Fungal Origin
por: Thai Le, Son, et al.
Publicado: (2019)

Dataset on structure, stability and myocardial effects of a new hybrid aspirin containing nitrogen monoxide-releasing molsidomine moiety
por: Szőke, Kitti, et al.
Publicado: (2019)

Nucleoside analogs for management of respiratory virus infections: mechanism of action and clinical efficacy
por: Stevaert, Annelies, et al.
Publicado: (2022)

Two Novel Semisynthetic Lipoglycopeptides Active against Staphylococcus aureus Biofilms and Cells in Late Stationary Growth Phase
por: Vimberg, Vladimir, et al.
Publicado: (2021)

Stereoselective Synthesis of Carbon-Sulfur-Bridged Glycomimetics by Photoinitiated Thiol-Ene Coupling Reactions
por: Csávás, Magdolna, et al.
Publicado: (2020)

Synthesis of β-d-galactopyranoside-Presenting Glycoclusters, Investigation of Their Interactions with Pseudomonas aeruginosa Lectin A (PA-IL) and Evaluation of Their Anti-Adhesion Potential
por: Malinovská, Lenka, et al.
Publicado: (2019)

Stereoselective Thioconjugation by Photoinduced Thiol‐ene Coupling Reactions of Hexo‐ and Pentopyranosyl d‐ and l‐Glycals at Low‐Temperature—Reactivity and Stereoselectivity Study
por: Kelemen, Viktor, et al.
Publicado: (2019)

Impact of SARS-CoV-2 Spike Mutations on Its Activation by TMPRSS2 and the Alternative TMPRSS13 Protease
por: Stevaert, Annelies, et al.
Publicado: (2022)

A Fucosylated Lactose-Presenting Tetravalent Glycocluster Acting as a Mutual Ligand of Pseudomonas aeruginosa Lectins A (PA-IL) and B (PA-IIL)—Synthesis and Interaction Studies
por: Csávás, Magdolna, et al.
Publicado: (2022)

N-acylhydrazone inhibitors of influenza virus PA endonuclease with versatile metal binding modes
por: Carcelli, Mauro, et al.
Publicado: (2016)

Synthesis of Tetravalent Thio- and Selenogalactoside-Presenting Galactoclusters and Their Interactions with Bacterial Lectin PA-IL from Pseudomonas aeruginosa
por: Illyés, Tünde Zita, et al.
Publicado: (2021)

Synthesis and Anticancer and Antiviral Activities of C-2′-Branched Arabinonucleosides
por: Bege, Miklós, et al.
Publicado: (2022)

Natural Apocarotenoids and Their Synthetic Glycopeptide Conjugates Inhibit SARS-CoV-2 Replication
por: Bereczki, Ilona, et al.
Publicado: (2021)

Novel Polymyxin-Inspired Peptidomimetics Targeting the SARS-CoV-2 Spike:hACE2 Interface
por: Bugatti, Kelly, et al.
Publicado: (2023)

Role of the viral hemagglutinin in the anti-influenza virus activity of newly synthesized polycyclic amine compounds
por: Torres, Eva, et al.
Publicado: (2013)

Favipiravir Does Not Inhibit Chikungunya Virus Replication in Mosquito Cells and Aedes aegypti Mosquitoes
por: Jacobs, Sofie, et al.
Publicado: (2021)

Teicoplanin pharmacokinetics during albumin dialysis
por: Weiler, Stefan, et al.
Publicado: (2010)

Is Therapeutic Drug Monitoring of Teicoplanin Useful?
por: Kim, Shin-Woo
Publicado: (2014)

Bacterial Cell Wall Analogue Peptides Control the Oligomeric States and Activity of the Glycopeptide Antibiotic Eremomycin: Solution NMR and Antimicrobial Studies
por: Izsépi, László, et al.
Publicado: (2021)

In vitro and in vivo antiplasmodial evaluation of sugar-modified nucleoside analogues
por: Bege, Miklós, et al.
Publicado: (2023)

Therapeutic Drug Concentrations of Teicoplanin in Clinical Settings
por: Nah, So-Yun, et al.
Publicado: (2014)

Tools for the Individualized Therapy of Teicoplanin for Neonates and Children
por: Ramos-Martín, V., et al.
Publicado: (2017)

Teicoplanin: an alternative drug for the treatment of COVID-19?
por: Baron, Sophie Alexandra, et al.
Publicado: (2020)

Clinical outcomes of teicoplanin use in the OPAT setting
por: Dabrowski, Hannah, et al.
Publicado: (2020)

The SARS-CoV-2 and other human coronavirus spike proteins are fine-tuned towards temperature and proteases of the human airways
por: Laporte, Manon, et al.
Publicado: (2021)

Basic Pharmacological Characterization of EV-34, a New H(2)S-Releasing Ibuprofen Derivative
por: Gyöngyösi, Alexandra, et al.
Publicado: (2021)

A Versatile Class of 1,4,4-Trisubstituted Piperidines Block Coronavirus Replication In Vitro
por: De Castro, Sonia, et al.
Publicado: (2022)

A Case of Hypersensitivity Syndrome to Both Vancomycin and Teicoplanin
por: Kwon, Hyouk-Soo, et al.
Publicado: (2006)

An Analogue of the Antibiotic Teicoplanin Prevents Flavivirus Entry In Vitro
por: De Burghgraeve, Tine, et al.
Publicado: (2012)

Pharmacokinetic/pharmacodynamic analysis of teicoplanin in patients with MRSA infections
por: Matsumoto, Kazuaki, et al.
Publicado: (2016)

Cannot write session to /tmp/vufind_sessions/sess_tt0cgglj5mfrkfs3ntn8sr28an