Cargando…

Design, synthesis, and biological evaluation of novel iso-d-2′,3′-dideoxy-3′-fluorothianucleoside derivatives

Novel iso-d-2′,3′-dideoxythianucleoside derivatives 1–4 were designed and asymmetrically synthesized as a bioisostere of lamivudine to search for new anti-HIV agents. The information about using sulfur participation occurred on DAST fluorination and Mitsunobu reaction will be of great help in synthe...

Descripción completa

Detalles Bibliográficos
Autores principales:	Kim, Kyung Ran, Moon, Hyung Ryong, Park, Ah-Young, Chun, Moon Woo, Jeong, Lak Shin
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Elsevier Ltd. 2007
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7127805/ https://www.ncbi.nlm.nih.gov/pubmed/17046264 http://dx.doi.org/10.1016/j.bmc.2006.09.066

Ejemplares similares

Dideoxy fluoro-ketopyranosyl nucleosides as potent antiviral agents: Synthesis and biological evaluation of 2,3- and 3,4-dideoxy-3-fluoro-4- and -2-keto-β-d-glucopyranosyl derivatives of N(4)-benzoyl cytosine
por: Manta, Stella, et al.
Publicado: (2009)

2-N-Benzyl-2,6-dideoxy-2,6-imino-3,4-O-isopropylidene-d-allononitrile
por: Ayers, Benjamin J., et al.
Publicado: (2013)

Creation of a Long-Acting Nanoformulated 2′,3′-Dideoxy-3′-Thiacytidine
por: Guo, Dongwei, et al.
Publicado: (2017)

N-Benzyl-1,3-dideoxy-1,3-imino-l-xylitol
por: Jenkinson, Sarah F., et al.
Publicado: (2011)

A Survey of Recent Synthetic Applications of 2,3-Dideoxy-Hex-2-enopyranosides
por: Gomez, Ana M., et al.
Publicado: (2015)

Design, synthesis, and antimelanogenic effects of (2-substituted phenyl-1,3-dithiolan-4-yl)methanol derivatives
por: Kim, Do Hyun, et al.
Publicado: (2017)

Design, synthesis, and biological evaluation of novel iso-flavones derivatives as H(3)R antagonists
por: Xin, Jian, et al.
Publicado: (2018)

Green synthesis of 1,5-dideoxy-1,5-imino-ribitol and 1,5-dideoxy-1,5-imino-dl-arabinitol from natural d-sugars over Au/Al(2)O(3) and SO(4)(2−)/Al(2)O(3) catalysts
por: Gao, Hongjian, et al.
Publicado: (2021)

(−)-Benzyl 2,3-dideoxy-β-d-erythro-hex-2-enopyranoside
por: Ohba, Shigeru, et al.
Publicado: (2013)

Synthesis and Biological Activity of 2′,3′-iso-Aryl-abscisic Acid Analogs
por: Wan, Chuan, et al.
Publicado: (2017)

Synthesis of enantiomerically pure d- and l-bicyclo[3.1.0]hexenyl carbanucleosides and their antiviral evaluation
por: Park, Ah-Young, et al.
Publicado: (2011)

Iso-seco-tanapartholides: Isolation, Synthesis and Biological Evaluation
por: Makiyi, Edward F, et al.
Publicado: (2009)

N-Benzyl-3,5-dideoxy-3,5-imino-1,2-O-isopropylidene-β-l-lyxofuranose
por: Edgeley, David S., et al.
Publicado: (2012)

Fluorine effect in nucleophilic fluorination at C4 of 1,6-anhydro-2,3-dideoxy-2,3-difluoro-β-D-hexopyranose
por: Lainé, Danny, et al.
Publicado: (2020)

Design, synthesis, and anti-melanogenic effects of (E)-2-benzoyl-3-(substituted phenyl)acrylonitriles
por: Yun, Hwi Young, et al.
Publicado: (2015)

2,6-Dideoxy-2,6-imino-l-glycero-d-ido-heptitol
por: Jenkinson, Sarah F., et al.
Publicado: (2009)

3-O-Benzhydryl-2,5-dideoxy-2,5-imino-2-C-methyl-l-lyxono-1,4-lactone
por: da Cruz, Filipa P., et al.
Publicado: (2008)

2-N-Benzyl-2,6-dideoxy-2,6-imino-3,4-O-isopropylidene-3-C-methyl-d-allononitrile
por: Ayers, Benjamin J., et al.
Publicado: (2012)

Dilute-‘N’-Go dideoxy sequencing of all DNA strands generated in multiplex LATE-PCR assays
por: Jia, Yanwei, et al.
Publicado: (2010)

Synthesis and Biological Evaluation of RGD and isoDGR–Monomethyl Auristatin Conjugates Targeting Integrin α(V)β(3)
por: Raposo Moreira Dias, André, et al.
Publicado: (2019)

Phenyl 4,6-di-O-acetyl-2,3-dideoxy-1-thio-α-d-erythro-hex-2-enopyranoside
por: Kinfe, Henok H., et al.
Publicado: (2011)

Design and Synthesis of 2,6-Disubstituted-4′-Selenoadenosine-5′-N,N-Dimethyluronamide Derivatives as Human A(3) Adenosine Receptor Antagonists
por: Choi, Hongseok, et al.
Publicado: (2021)

Total Synthesis of Resveratrone and iso‐Resveratrone
por: Fritsch, Stefan, et al.
Publicado: (2022)

Cross-resistance studies on 1,6-dibromo-dideoxy-D-mannitol(DBM)-resistant Yoshida S.C. sarcoma.
por: Csányi, E., et al.
Publicado: (1967)

Rapid, effective and low-cost purification of dideoxy-sequencing reactions by home-made magnetic beads suspension and magnetic separator
por: Sassa, Hidenori, et al.
Publicado: (2022)

Design and Synthesis of (Z)-5-(Substituted benzylidene)-3-cyclohexyl-2-thioxothiazolidin-4-one Analogues as Anti-Tyrosinase and Antioxidant Compounds: In Vitro and In Silico Insights
por: Ko, Jeongin, et al.
Publicado: (2022)

Monoclinic polymorph of 2,5-dideoxy-2,5-epithio-1,3:4,6-bis-O-[(R)-phenylmethylene]-l-iditol
por: Gibson, Jerrell G., et al.
Publicado: (2012)

Synthesis and Biological Screening of New Cyano-Substituted Pyrrole Fused (Iso)Quinoline Derivatives
por: Al-Matarneh, Maria Cristina, et al.
Publicado: (2021)

Technical product documentation: Part 3: applications of ISO-13567-1 and ISO-13567-2
por: International Organization for Standardization. Geneva
Publicado: (1999)

Beam Characterization of Linac 4's ISO3
por: Noll, Daniel, et al.
Publicado: (2019)

Prop-2-yn-1-yl 4,6-di-O-acetyl-2,3-dideoxy-α-d-erythro-hex-2-enopyranoside
por: Mesfin, Fanuel M., et al.
Publicado: (2011)

ISO 14000 - ISO 9000
por: Rothery, Brian

Synthesis and biological evaluation of RGD and isoDGR peptidomimetic-α-amanitin conjugates for tumor-targeting
por: Bodero, Lizeth, et al.
Publicado: (2018)

Tumour-inhibiting Action of 1,6-Di-(2-Bromoethylamino)-1,6-Dideoxy-D-Mannitol Dihydrobromide [DBM (R13)]
por: Baló, J., et al.
Publicado: (1959)

ISO 9001 for engineers and designers
por: Schoonmaker, Stephen J.
Publicado: (1996)

Design, Synthesis, In Vitro, and In Silico Insights of 5-(Substituted benzylidene)-2-phenylthiazol-4(5H)-one Derivatives: A Novel Class of Anti-Melanogenic Compounds
por: Yoon, Dahye, et al.
Publicado: (2023)

Total Synthesis of (+)-Petromyroxol, (−)-iso-Petromyroxol, and Possible Diastereomers
por: Mullapudi, Venkannababu, et al.
Publicado: (2020)

Open Design 3D-Printable Adjustable Micropipette that Meets the ISO Standard for Accuracy
por: Brennan, Martin D., et al.
Publicado: (2018)

Design and Synthesis of (Z)-2-(Benzylamino)-5-benzylidenethiazol-4(5H)-one Derivatives as Tyrosinase Inhibitors and Their Anti-Melanogenic and Antioxidant Effects
por: Lee, Jieun, et al.
Publicado: (2023)

Synthesis and crystal structure of (E)-2-benzyl-1,3-diphenylisothiouronium iodide
por: Kang, Sungmin, et al.
Publicado: (2022)

Cannot write session to /tmp/vufind_sessions/sess_5pn408iose0mcfl61j3rgbt7cl