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Synthesis, Characterization and Biological Evaluation of Novel Dihydropyranoindoles Improving the Anticancer Effects of HDAC Inhibitors
The dihydropyranoindole scaffold was identified as a promising target for improving the anti-cancer activity of HDAC inhibitors from the preliminary screening of a library of compounds. A suitable methodology has been developed for the preparation of novel dihydropyranoindoles via the Hemetsberger i...
Autores principales: | Bingul, Murat, Arndt, Greg M., Marshall, Glenn M., Cheung, Belamy B., Kumar, Naresh, Black, David StC. |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
MDPI
2020
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7144403/ https://www.ncbi.nlm.nih.gov/pubmed/32197360 http://dx.doi.org/10.3390/molecules25061377 |
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