Cascade trifluoromethylthiolation and cyclization of N-[(3-aryl)propioloyl]indoles

A cascade oxidative trifluoromethylthiolation and cyclization of N-[(3-aryl)propioloyl]indoles with AgSCF(3) is described. This protocol allows for the synthesis of novel bis(trifluoromethylthiolated) or trifluoromethylthiolated pyrrolo[1,2-a]indol-3-ones in moderate to good yields. Mechanistic inve...

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Detalles Bibliográficos
Autores principales: Bi, Ming-Xi, Liu, Shuai, Huang, Yangen, Xu, Xiu-Hua, Qing, Feng-Ling
Formato: Online Artículo Texto
Lenguaje:English
Publicado: Beilstein-Institut 2020
Materias:
Letter
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7155893/
https://www.ncbi.nlm.nih.gov/pubmed/32318122
http://dx.doi.org/10.3762/bjoc.16.62

Internet

https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7155893/
https://www.ncbi.nlm.nih.gov/pubmed/32318122
http://dx.doi.org/10.3762/bjoc.16.62

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