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Fluorescent analogues of BeKm-1 with high and specific activity against the hERG channel
Peptidic toxins that target specifically mammalian channels and receptors can be found in the venom of animals. These toxins are rarely used directly as tools for biochemical experiments, and need to be modified via the attachment of chemical groups (e.g., radioactive or fluorescent moieties). Ideal...
Autores principales: | Vasseur, Lucie, Chavanieu, Alain, Combemale, Stéphanie, Caumes, Cécile, Béroud, Rémy, De Waard, Michel, Ducrot, Pierre, Boutin, Jean A., Ferry, Gilles, Cens, Thierry |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Elsevier
2019
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7285999/ https://www.ncbi.nlm.nih.gov/pubmed/32550567 http://dx.doi.org/10.1016/j.toxcx.2019.100010 |
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