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Synthesis and biological evaluation of novel quinoline-piperidine scaffolds as antiplasmodium agents
The parasitic disease malaria places almost half of the world’s population at risk of infection and is responsible for more than 400,000 deaths each year. The first-line treatment, artemisinin combination therapies (ACT) regimen, is under threat due to emerging resistance of Plasmodium falciparum st...
Autores principales: | Van de Walle, Tim, Boone, Maya, Van Puyvelde, Julie, Combrinck, Jill, Smith, Peter J., Chibale, Kelly, Mangelinckx, Sven, D’hooghe, Matthias |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Editions Scientifiques Elsevier
2020
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7294232/ https://www.ncbi.nlm.nih.gov/pubmed/32408064 http://dx.doi.org/10.1016/j.ejmech.2020.112330 |
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