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Activation of μ‐opioid receptors by MT‐45 (1‐cyclohexyl‐4‐(1,2‐diphenylethyl)piperazine) and its fluorinated derivatives
BACKGROUND AND PURPOSE: A fluorinated derivative (2F‐MT‐45) of the synthetic μ‐opioid receptor agonist MT‐45 (1‐cyclohexyl‐4‐(1,2‐diphenylethyl)piperazine) was recently identified in a seized illicit tablet. While MT‐45 is a Class A drug, banned in a number of countries, nothing is known about the p...
Autores principales: | Baptista‐Hon, Daniel T., Smith, Mark, Singleton, Samuel, Antonides, Lysbeth H., Nic Daeid, Niamh, McKenzie, Craig, Hales, Tim G. |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
John Wiley and Sons Inc.
2020
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7348096/ https://www.ncbi.nlm.nih.gov/pubmed/32246840 http://dx.doi.org/10.1111/bph.15064 |
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