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Structure-Activity Relationships for the Anaesthetic and Analgaesic Properties of Aromatic Ring-Substituted Ketamine Esters
A series of benzene ring substituted ketamine N-alkyl esters were prepared from the corresponding substituted norketamines. Few of the latter have been reported since they have not been generally accessible via known routes. We report a new general route to many of these norketamines via the Neber (...
Autores principales: | Dimitrov, Ivaylo V., Harvey, Martyn G., Voss, Logan J., Sleigh, James W., Bickerdike, Michael J., Denny, William A. |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
MDPI
2020
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7356787/ https://www.ncbi.nlm.nih.gov/pubmed/32604891 http://dx.doi.org/10.3390/molecules25122950 |
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