Synthesis and evaluation of 2,4,5-trisubstitutedthiazoles as carbonic anhydrase-III inhibitors

A series of 17 compounds (12–16 b) with 2,4,5-trisubstitutedthiazole scaffold having 5-aryl group, 4-carboxylic acid/ester moiety, and 2-amino/amido/ureido functional groups were synthesised, characterised, and evaluated for their carbonic anhydrase (CA)-III inhibitory activities using the size excl...

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Detalles Bibliográficos
Autores principales: Al-Jaidi, Bilal A., Deb, Pran Kishore, Telfah, Soha Taher, Dakkah, Abdel Naser, Bataineh, Yazan A., Khames Aga, Qutaiba Ahmed Al, Al-dhoun, Mohammad A., Ahmad Al-Subeihi, Ala’ Ali, Odetallah, Haifa’a Marouf, Bardaweel, Sanaa K., Mailavaram, Raghuprasad, Venugopala, Katharigatta N., Nair, Anroop B.
Formato: Online Artículo Texto
Lenguaje:English
Publicado: Taylor & Francis 2020
Materias:
Original Article
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7470151/
https://www.ncbi.nlm.nih.gov/pubmed/32635773
http://dx.doi.org/10.1080/14756366.2020.1786820

Internet

https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7470151/
https://www.ncbi.nlm.nih.gov/pubmed/32635773
http://dx.doi.org/10.1080/14756366.2020.1786820

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