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Vitamin B3-Based Biologically Active Compounds as Inhibitors of Human Cholinesterases
We evaluated the potential of nine vitamin B3 scaffold-based derivatives as acetylcholinesterase (AChE) and butyrylcholinesterase (BChE) inhibitors, as a starting point for the development of novel drugs for treating disorders with cholinergic neurotransmission-linked pathology. As the results indic...
Autores principales: | Zandona, Antonio, Lihtar, Gabriela, Maraković, Nikola, Miš, Katarina, Bušić, Valentina, Gašo-Sokač, Dajana, Pirkmajer, Sergej, Katalinić, Maja |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
MDPI
2020
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7663184/ https://www.ncbi.nlm.nih.gov/pubmed/33138280 http://dx.doi.org/10.3390/ijms21218088 |
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