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Insights into the Membranolytic Activity of Antimalarial Drug-Cell Penetrating Peptide Conjugates

Conjugation of TP10, a cell-penetrating peptide with intrinsic antimalarial activity, to the well-known antimalarial drugs chloroquine and primaquine has been previously shown to enhance the peptide’s action against, respectively, blood- and liver-stage malaria parasites. Yet, this was achieved at t...

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Detalles Bibliográficos
Autores principales:	Aguiar, Luísa, Pinheiro, Marina, Neves, Ana Rute, Vale, Nuno, Defaus, Sira, Andreu, David, Reis, Salette, Gomes, Paula
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2020
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7822033/ https://www.ncbi.nlm.nih.gov/pubmed/33375073 http://dx.doi.org/10.3390/membranes11010004

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