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2-Chloro-3-nitro-5-(trifluoromethyl)benzoic acid and -benzamide: structural characterization of two precursors for antitubercular benzothiazinones

8-Nitro-1,3-benzothiazin-4-ones are a promising class of new antitubercular agents, two candidates of which, namely BTZ043 and PBTZ169 (INN: macozinone), have reached clinical trials. The crystal and molecular structures of two synthetic precursors, 2-chloro-3-nitro-5-(trifluoromethyl)benzoic...

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Detalles Bibliográficos
Autores principales:	Richter, Adrian, Goddard, Richard, Schlegel, Tom, Imming, Peter, Seidel, Rüdiger W.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	International Union of Crystallography 2021
Materias:	Research Communications
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7869535/ https://www.ncbi.nlm.nih.gov/pubmed/33614143 http://dx.doi.org/10.1107/S2056989021000517

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