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Occurrence of Morpholine in Central Nervous System Drug Discovery
[Image: see text] Developing drugs for the central nervous system (CNS) requires fine chemical modifications, as a strict balance between size and lipophilicity is necessary to improve the permeability through the blood-brain barrier (BBB). In this context, morpholine and its analogues represent val...
Autores principales: | Lenci, Elena, Calugi, Lorenzo, Trabocchi, Andrea |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
American Chemical
Society
2021
|
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7877733/ https://www.ncbi.nlm.nih.gov/pubmed/33459557 http://dx.doi.org/10.1021/acschemneuro.0c00729 |
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