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Computational Modeling to Explain Why 5,5-Diarylpentadienamides are TRPV1 Antagonists

Several years ago, the crystallographic structures of the transient receptor potential vanilloid 1 (TRPV1) in the presence of agonists and antagonists were reported, providing structural information about its chemical activation and inactivation. TRPV1’s activation increases the transport of calcium...

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Detalles Bibliográficos
Autor principal:	Caballero, Julio
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2021
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8004144/ https://www.ncbi.nlm.nih.gov/pubmed/33801115 http://dx.doi.org/10.3390/molecules26061765

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