Cargando…
Novel Pyrimidine Derivatives as Potential Anticancer Agents: Synthesis, Biological Evaluation and Molecular Docking Study
In the present paper, new pyrimidine derivatives were designed, synthesized and analyzed in terms of their anticancer properties. The tested compounds were evaluated in vitro for their antitumor activity. The cytotoxic effect on normal human dermal fibroblasts (NHDF) was also determined. According t...
Autores principales: | Tylińska, Beata, Wiatrak, Benita, Czyżnikowska, Żaneta, Cieśla-Niechwiadowicz, Aneta, Gębarowska, Elżbieta, Janicka-Kłos, Anna |
---|---|
Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
MDPI
2021
|
Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8067809/ https://www.ncbi.nlm.nih.gov/pubmed/33917090 http://dx.doi.org/10.3390/ijms22083825 |
Ejemplares similares
-
New Oxazolo[5,4-d]pyrimidines as Potential Anticancer Agents: Their Design, Synthesis, and In Vitro Biological Activity Research
por: Sochacka-Ćwikła, Aleksandra, et al.
Publicado: (2022) -
Design and Synthesis of N-Substituted 3,4-Pyrroledicarboximides as Potential Anti-Inflammatory Agents
por: Redzicka, Aleksandra, et al.
Publicado: (2021) -
Design, Synthesis, Biological Evaluation, and Molecular Docking Study of 4,6-Dimethyl-5-aryl/alkyl-2-[2-hydroxy-3-(4-substituted-1-piperazinyl)propyl]pyrrolo[3,4-c]pyrrole-1,3(2H,5H)-diones as Anti-Inflammatory Agents with Dual Inhibition of COX and LOX
por: Redzicka, Aleksandra, et al.
Publicado: (2023) -
Bioactive Olivacine Derivatives—Potential Application in Cancer Therapy
por: Tylińska, Beata, et al.
Publicado: (2021) -
Synthesis of New Tricyclic 1,2-Thiazine Derivatives with Anti-Inflammatory Activity
por: Maniewska, Jadwiga, et al.
Publicado: (2021)