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A Class of Valuable (Pro-)Activity-Based Protein Profiling Probes: Application to the Redox-Active Antiplasmodial Agent, Plasmodione

[Image: see text] Plasmodione (PD) is a potent antimalarial redox-active drug acting at low nM range concentrations on different malaria parasite stages. In this study, in order to determine the precise PD protein interactome in parasites, we developed a class of (pro-)activity-based protein profili...

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Detalles Bibliográficos
Autores principales: Cichocki, Bogdan Adam, Khobragade, Vrushali, Donzel, Maxime, Cotos, Leandro, Blandin, Stephanie, Schaeffer-Reiss, Christine, Cianférani, Sarah, Strub, Jean-Marc, Elhabiri, Mourad, Davioud-Charvet, Elisabeth
Formato: Online Artículo Texto
Lenguaje:English
Publicado: American Chemical Society 2021
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8154199/
https://www.ncbi.nlm.nih.gov/pubmed/34056636
http://dx.doi.org/10.1021/jacsau.1c00025