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Pyrimidin‐6‐yl Trifluoroborate Salts as Versatile Templates for Heterocycle Synthesis
We report a novel and general method to access a highly under‐studied privileged scaffold—pyrimidines bearing a trifluoroborate at C4, and highlight the broad utility of these intermediates in a rich array of downstream functionalization reactions. This chemistry is underpinned by the unique feature...
Autores principales: | Cousins, David L., Fricero, Prisca, Kopf, Kenji P. M., McColl, Elliot J., Czechtizky, Werngard, Lim, Yee Hwee, Harrity, Joseph P. A. |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
John Wiley and Sons Inc.
2021
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8252621/ https://www.ncbi.nlm.nih.gov/pubmed/33570831 http://dx.doi.org/10.1002/anie.202101297 |
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