Tritylamine as an Ammonia Surrogate in the Ugi Reaction Provides Access to Unprecedented 5-Sulfamido Oxazoles Using Burgess-type Reagents

[Image: see text] Starting from a wide range of α-acylamino amide substructures synthesized using tritylamine as an ammonia surrogate in the Ugi reaction, Burgess-type reagents enable cyclodehydration and afford unprecedented oxazole scaffolds with four points of diversity, including a sulfamide moi...

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Detalles Bibliográficos
Autores principales: Bhela, Irene Preet, Serafini, Marta, Del Grosso, Erika, Tron, Gian Cesare, Pirali, Tracey
Formato: Online Artículo Texto
Lenguaje:English
Publicado: American Chemical Society 2021
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8289289/
https://www.ncbi.nlm.nih.gov/pubmed/33913716
http://dx.doi.org/10.1021/acs.orglett.1c01002

Internet

https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8289289/
https://www.ncbi.nlm.nih.gov/pubmed/33913716
http://dx.doi.org/10.1021/acs.orglett.1c01002

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