Cargando…
The selectivity of α‐adrenoceptor agonists for the human α1A, α1B, and α1D‐adrenoceptors
Highly selective drugs offer a way to minimize side‐effects. For agonist ligands, this could be through highly selective affinity or highly selective efficacy, but this requires careful measurements of intrinsic efficacy. The α1‐adrenoceptors are important clinical targets, and α1‐agonists are used...
| Autores principales: | , |
|---|---|
| Formato: | Online Artículo Texto |
| Lenguaje: | English |
| Publicado: |
John Wiley and Sons Inc.
2021
|
| Materias: | |
| Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8343220/ https://www.ncbi.nlm.nih.gov/pubmed/34355529 http://dx.doi.org/10.1002/prp2.799 |