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Determination of the Absolute Configuration of Bioactive Indole-Containing Pyrazino[2,1-b]quinazoline-3,6-diones and Study of Their In Vitro Metabolic Profile
In recent decades, fungi-derived naturally occurring quinazolines have emerged as potential drug candidates. Nevertheless, most studies are conducted for bioactivity assays, and little is known about their absorption, distribution, metabolism, and elimination (ADME) properties. To perform metabolic...
Autores principales: | Long, Solida, Furlani, Izadora L., de Oliveira, Juliana M., Resende, Diana I. S. P., Silva, Artur M. S., Gales, Luís, Pereira, José A., Kijjoa, Anake, Cass, Quezia B., Oliveira, Regina V., Sousa, Emília, Pinto, Madalena M. M. |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
MDPI
2021
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8398919/ https://www.ncbi.nlm.nih.gov/pubmed/34443658 http://dx.doi.org/10.3390/molecules26165070 |
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