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Selective Recognition of a Single HIV-1 G-Quadruplex by Ultrafast Small-Molecule Screening

[Image: see text] G-quadruplexes (G4s) are implicated in pathological processes such as cancer and infective diseases. Their targeting with G4-ligands has shown therapeutic capacity. Most of the current G4-ligands are planar molecules, do not discriminate among G4s, and have poor druglike properties...

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Detalles Bibliográficos
Autores principales: Scalabrin, Matteo, Nadai, Matteo, Tassinari, Martina, Lago, Sara, Doria, Filippo, Frasson, Ilaria, Freccero, Mauro, Richter, Sara N.
Formato: Online Artículo Texto
Lenguaje:English
Publicado: American Chemical Society 2021
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8613737/
https://www.ncbi.nlm.nih.gov/pubmed/34762806
http://dx.doi.org/10.1021/acs.analchem.0c04106