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A Phenylfurocoumarin Derivative Reverses ABCG2-Mediated Multidrug Resistance In Vitro and In Vivo

The ATP-binding cassette subfamily G member 2 (ABCG2) transporter is involved in the development of multidrug resistance in cancer patients. Many inhibitors of ABCG2 have been reported to enhance the chemosensitivity of cancer cells. However, none of these inhibitors are being used clinically. The a...

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Detalles Bibliográficos
Autores principales: Kokubo, Shoji, Ohnuma, Shinobu, Murakami, Megumi, Kikuchi, Haruhisa, Funayama, Shota, Suzuki, Hideyuki, Kajiwara, Taiki, Yamamura, Akihiro, Karasawa, Hideaki, Sugisawa, Norihiko, Ohsawa, Kosuke, Kano, Kuniyuki, Aoki, Junken, Doi, Takayuki, Naitoh, Takeshi, Ambudkar, Suresh V., Unno, Michiaki
Formato: Online Artículo Texto
Lenguaje:English
Publicado: MDPI 2021
Materias:
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8618058/
https://www.ncbi.nlm.nih.gov/pubmed/34830383
http://dx.doi.org/10.3390/ijms222212502