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New Compounds with Bioisosteric Replacement of Classic Choline Kinase Inhibitors Show Potent Antiplasmodial Activity
In the fight against Malaria, new strategies need to be developed to avoid resistance of the parasite to pharmaceutics and other prevention barriers. Recently, a Host Directed Therapy approach based on the suppression of the starting materials uptake from the host by the parasite has provided excell...
Autores principales: | Aguilar-Troyano, Francisco José, Torretta, Archimede, Rubbini, Gianluca, Fasiolo, Alberto, Luque-Navarro, Pilar María, Carrasco-Jimenez, María Paz, Pérez-Moreno, Guiomar, Bosch-Navarrete, Cristina, González-Pacanowska, Dolores, Parisini, Emilio, Lopez-Cara, Luisa Carlota |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
MDPI
2021
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8621770/ https://www.ncbi.nlm.nih.gov/pubmed/34834257 http://dx.doi.org/10.3390/pharmaceutics13111842 |
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