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Synthesis of Azacarbolines via PhIO(2)-Promoted Intramolecular Oxidative Cyclization of α-Indolylhydrazones
[Image: see text] An unprecedented synthesis of polysubstituted indole-fused pyridazines (azacarbolines) from α-indolylhydrazones under oxidative conditions using a combination of iodylbenzene (PhIO(2)) and trifluoroacetic acid (TFA) has been developed. This transformation is conducted without the n...
Autores principales: | , , , , , |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
American Chemical Society
2021
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Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8689645/ https://www.ncbi.nlm.nih.gov/pubmed/34871002 http://dx.doi.org/10.1021/acs.joc.1c02217 |