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Radiosensitizing effect of c-Met kinase inhibitor BPI-9016M in esophageal squamous cell carcinoma cells in vitro and in vivo

BACKGROUND: c-Met is the receptor of hepatocyte growth factor (HGF) which plays a key role in inhibiting apoptosis. BPI-9016M is a small-molecule c-Met inhibitor that can promote apoptosis and enhance the cytotoxicity of various DNA-damaging agents. Here, we evaluated the radiosensitizing potential...

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Detalles Bibliográficos
Autores principales: Jiang, Chenxue, Han, Shuiyun, Sun, Xiaojiang, Xu, Yaping, Feng, Jianguo, Shang, Jinbiao
Formato: Online Artículo Texto
Lenguaje:English
Publicado: AME Publishing Company 2021
Materias:
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8756247/
https://www.ncbi.nlm.nih.gov/pubmed/35071493
http://dx.doi.org/10.21037/atm-21-6586