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Self-Assembled Micellar Glutaminase Allosteric Inhibitor for Effective Therapeutic Intervention

INTRODUCTION: Kidney-type glutaminase (KGA) has been an important anti-tumor drug target, and KGA allosteric inhibitors attracted much interest for their superior enzymatic specificity with good drug safety profiles. For glutaminase allosteric inhibitors such as BPTES, CB-839 and Selen derivatives,...

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Detalles Bibliográficos
Autores principales:	Fang, Jinzhang, Chen, Zhao, Li, Jinxiu, Li, Di, Wang, Wenxi, Ruan, Benfang Helen
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Dove 2022
Materias:	Original Research
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8764296/ https://www.ncbi.nlm.nih.gov/pubmed/35058693 http://dx.doi.org/10.2147/IJN.S346596

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