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Effect of Ions and Sequence Variants on the Antagonist Binding Properties of the Histamine H(1) Receptor
The histamine H(1) receptor (H(1)R) is a G protein-coupled receptor (GPCR) and represents a main target in the treatment of allergic reactions as well as inflammatory reactions and depressions. Although the overall effect of antagonists on H(1) function has been extensively investigated, rather litt...
Autores principales: | Conrad, Marcus, Söldner, Christian A., Sticht, Heinrich |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
MDPI
2022
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8836275/ https://www.ncbi.nlm.nih.gov/pubmed/35163341 http://dx.doi.org/10.3390/ijms23031420 |
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