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Design, Synthesis, and Biological Evaluation of 4,4’-Difluorobenzhydrol Carbamates as Selective M(1) Antagonists
Due to their important role in mediating a broad range of physiological functions, muscarinic acetylcholine receptors (mAChRs) have been a promising target for therapeutic and diagnostic applications alike; however, the list of truly subtype-selective ligands is scarce. Within this work, we have ide...
Autores principales: | Kilian, Jonas, Ozenil, Marius, Millard, Marlon, Fürtös, Dorka, Maisetschläger, Verena, Holzer, Wolfgang, Wadsak, Wolfgang, Hacker, Marcus, Langer, Thierry, Pichler, Verena |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
MDPI
2022
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8879200/ https://www.ncbi.nlm.nih.gov/pubmed/35215360 http://dx.doi.org/10.3390/ph15020248 |
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