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Design, Synthesis, and Evaluation of Novel 2H-Benzo[b][1,4]thiazin-3(4H)-one Derivatives as New Acetylcholinesterase Inhibitors
Alzheimer’s disease (AD) is a slowly progressive neurodegenerative disease that causes dementia in people aged 65 and over. In the present study, a series of thiadiazole hybrid compounds with benzothiazine derivatives as acetylcholinesterase inhibitors were developed and evaluated for their biologic...
Autores principales: | Haji Ali, Sazan, Osmaniye, Derya, Sağlık, Begüm Nurpelin, Levent, Serkan, Özkay, Yusuf, Kaplancıklı, Zafer Asım |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
MDPI
2022
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9000418/ https://www.ncbi.nlm.nih.gov/pubmed/35408519 http://dx.doi.org/10.3390/molecules27072121 |
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