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Sequential ligand- and structure-based virtual screening approach for the identification of potential G protein-coupled estrogen receptor-1 (GPER-1) modulators

G protein-coupled estrogen receptor-1 (GPER-1) is a seven transmembrane receptor, responsible for mediating rapid estrogen signaling in many physiological responses in reproductive, nervous, endocrine, immune and cardiovascular systems. Due to unavailability of the crystal structure of GPER-1, we ha...

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Detalles Bibliográficos
Autores principales:	Khan, Shafi Ullah, Ahemad, Nafees, Chuah, Lay-Hong, Naidu, Rakesh, Htar, Thet Thet
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	The Royal Society of Chemistry 2019
Materias:	Chemistry
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9059856/ https://www.ncbi.nlm.nih.gov/pubmed/35520492 http://dx.doi.org/10.1039/c8ra09318k

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