Cargando…

An efficient 3-acylquinoline synthesis from acetophenones and anthranil via C(sp(3))–H bond activation mediated by Selectfluor

An efficient method for the synthesis of 3-functionalized quinolines from commercially available acetophenones and anthranil has been described. Selectfluor propels the C(sp(3))–H bond activation of the acetophenones and aza-Michael addition of anthranil resulting in annulated 3-acylquinolines in mo...

Descripción completa

Detalles Bibliográficos
Autores principales: Gao, Yejun, Hider, Robert C., Ma, Yongmin
Formato: Online Artículo Texto
Lenguaje:English
Publicado: The Royal Society of Chemistry 2019
Materias:
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9062302/
https://www.ncbi.nlm.nih.gov/pubmed/35520934
http://dx.doi.org/10.1039/c9ra01481k