Synthesis of 2-BMIDA Indoles via Heteroannulation: Applications in Drug Scaffold and Natural Product Synthesis

[Image: see text] A Pd-catalyzed heteroannulation approach for the synthesis of C2 borylated indoles is reported. The process allows access to highly functionalized 2-borylated indole scaffolds with complete control of regioselectivity. The utility of the process is demonstrated in the synthesis of...

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Detalles Bibliográficos
Autores principales: Bell, George E., Fyfe, James W. B., Israel, Eva M., Slawin, Alexandra M. Z., Campbell, Matthew, Watson, Allan J. B.
Formato: Online Artículo Texto
Lenguaje:English
Publicado: American Chemical Society 2022
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9062883/
https://www.ncbi.nlm.nih.gov/pubmed/35426314
http://dx.doi.org/10.1021/acs.orglett.2c00959

Internet

https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9062883/
https://www.ncbi.nlm.nih.gov/pubmed/35426314
http://dx.doi.org/10.1021/acs.orglett.2c00959

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